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Effect of verapamil on the pharmacokinetics of hydroxycamptothecin and its potential mechanism

CONTEXT: Hydroxycamptothecin (HCPT) has antitumor activity in various cancers, but its poor bioavailability and efflux limit its clinical application. Verapamil has been demonstrated to improve the bioavailability of many drugs. However, the effect of verapamil on the pharmacokinetics of HCPT was no...

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Опубликовано в: :Pharm Biol
Главные авторы: Xing, Hua, Luo, Xiao, Li, Yang, Fan, Chunni, Liu, Ning, Cui, Chunguo, Li, Wenjia
Формат: Artigo
Язык:Inglês
Опубликовано: Taylor & Francis 2020
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC7034088/
https://ncbi.nlm.nih.gov/pubmed/31990625
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1080/13880209.2020.1717550
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