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Application of hot melt extrusion to enhance the dissolution and oral bioavailability of oleanolic acid

The aim of this study was to improve the in vitro dissolution rate and oral bioavailability of oleanolic acid (OA), a water insoluble drug belonging to BCS class IV. Hot melt extrusion (HME) was applied to develop OA amorphous solid dispersions. The characterizations of the optimal formulation were...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Argitaratua izan da:Asian J Pharm Sci
Egile Nagusiak: Gao, Nannan, Guo, Mengran, Fu, Qiang, He, Zhonggui
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: Shenyang Pharmaceutical University 2017
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC7032251/
https://ncbi.nlm.nih.gov/pubmed/32104315
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ajps.2016.06.006
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