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Functionalized Naphthalimide-4-aminoquinoline Conjugates as Promising Antiplasmodials, with Mechanistic Insights

[Image: see text] A series of 25 conjugates has been synthesized to evaluate their antiplasmodial potency and cytotoxicity against the chloroquine resistant (CQR) W2 strain of P. falciparum and Vero kidney cell lines, respectively. Most of the compounds showed IC(50) values in the lower nM range and...

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Publicado en:ACS Med Chem Lett
Autores principales: Shalini, Legac, Jenny, Adeniyi, Adebayo A., Kisten, Prishani, Rosenthal, Philip J., Singh, Parvesh, Kumar, Vipan
Formato: Artigo
Lenguaje:Inglês
Publicado: American Chemical Society 2020
Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC7025377/
https://ncbi.nlm.nih.gov/pubmed/32071682
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsmedchemlett.9b00521
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