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Computer-Aided Design of Cefuroxime Axetil/Cyclodextrin System with Enhanced Solubility and Antimicrobial Activity

This study aimed to investigate changes in the solubility and antimicrobial efficacy of cefuroxime axetil (CA) when incorporated into cyclodextrin (CD). While choosing the CD, the validated in silico model was used. A theoretical model based on docking and molecular mechanics/generalized born surfac...

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Detalhes bibliográficos
Publicado no:Biomolecules
Main Authors: Mizera, Mikołaj, Szymanowska, Daria, Stasiłowicz, Anna, Siąkowska, Dominika, Lewandowska, Kornelia, Miklaszewski, Andrzej, Plech, Tomasz, Tykarska, Ewa, Cielecka-Piontek, Judyta
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2019
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7023374/
https://ncbi.nlm.nih.gov/pubmed/31878057
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/biom10010024
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