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Degradation of proteins by PROTACs and other strategies

Blocking the biological functions of scaffold proteins and aggregated proteins is a challenging goal. PROTAC proteolysis-targeting chimaera (PROTAC) technology may be the solution, considering its ability to selectively degrade target proteins. Recent progress in the PROTAC strategy include identifi...

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Publicat a:Acta Pharm Sin B
Autors principals: Wang, Yang, Jiang, Xueyang, Feng, Feng, Liu, Wenyuan, Sun, Haopeng
Format: Artigo
Idioma:Inglês
Publicat: Elsevier 2020
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7016280/
https://ncbi.nlm.nih.gov/pubmed/32082969
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.apsb.2019.08.001
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