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Gilteritinib induces PUMA‐dependent apoptotic cell death via AKT/GSK‐3β/NF‐κB pathway in colorectal cancer cells

As a highly potent and highly selective oral inhibitor of FLT3/AXL, gilteritinib showed activity against FLT3D835 and FLT3‐ITD mutations in pre‐clinical testing, although its role on colorectal cancer (CRC) cells is not yet fully elucidated. We examined the activity of gilteritinib in suppressing gr...

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Pubblicato in:J Cell Mol Med
Autori principali: Li, Liangjun, Lin, Lin, Li, Ming, Li, Weiling
Natura: Artigo
Lingua:Inglês
Pubblicazione: John Wiley and Sons Inc. 2019
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7011145/
https://ncbi.nlm.nih.gov/pubmed/31881122
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/jcmm.14913
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