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The functionally relevant site for paxilline inhibition of BK channels

The tremorgenic fungal alkaloid paxilline (PAX) is a commonly used specific inhibitor of the large-conductance, voltage- and Ca(2+)-dependent BK-type K(+) channel. PAX inhibits BK channels by selective interaction with closed states. BK inhibition by PAX is best characterized by the idea that PAX ga...

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Bibliographic Details
Published in:Proc Natl Acad Sci U S A
Main Authors: Zhou, Yu, Xia, Xiao-Ming, Lingle, Christopher J.
Format: Artigo
Language:Inglês
Published: National Academy of Sciences 2020
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Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC6969516/
https://ncbi.nlm.nih.gov/pubmed/31879339
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.1912623117
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