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Molecular dynamics simulations on RORγt: insights into its functional agonism and inverse agonism

The retinoic acid receptor-related orphan receptor (ROR) γt receptor is a member of nuclear receptors, which is indispensable for the expression of pro-inflammatory cytokine IL-17. RORγt has been established as a drug target to design and discover novel treatments for multiple inflammatory and immun...

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Dades bibliogràfiques
Publicat a:Acta Pharmacol Sin
Autors principals: Yuan, Cong-min, Chen, Hai-hong, Sun, Nan-nan, Ma, Xiao-jun, Xu, Jun, Fu, Wei
Format: Artigo
Idioma:Inglês
Publicat: Springer Singapore 2019
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6961238/
https://ncbi.nlm.nih.gov/pubmed/31316175
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41401-019-0259-z
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