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Direct and Indirect Quantification of Phosphate Metabolites of Nucleoside Analogs in Biological Samples

Nucleoside reverse transcriptase inhibitors (NRTIs) are prodrugs that require intracellular phosphorylation to active triphosphate nucleotide metabolites (NMs) for their pharmacological activity. However, monitoring these pharmacologically active NMs is challenging due to their instability, high hyd...

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Detalles Bibliográficos
Publicado en:J Pharm Biomed Anal
Autores principales: Gautam, Nagsen, Alamoudi, Jawaher Abdullah, Kumar, Sushil, Alnouti, Yazen
Formato: Artigo
Lenguaje:Inglês
Publicado: 2019
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC6931899/
https://ncbi.nlm.nih.gov/pubmed/31610397
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.jpba.2019.112902
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