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Direct and Indirect Quantification of Phosphate Metabolites of Nucleoside Analogs in Biological Samples

Nucleoside reverse transcriptase inhibitors (NRTIs) are prodrugs that require intracellular phosphorylation to active triphosphate nucleotide metabolites (NMs) for their pharmacological activity. However, monitoring these pharmacologically active NMs is challenging due to their instability, high hyd...

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Dettagli Bibliografici
Pubblicato in:J Pharm Biomed Anal
Autori principali: Gautam, Nagsen, Alamoudi, Jawaher Abdullah, Kumar, Sushil, Alnouti, Yazen
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2019
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6931899/
https://ncbi.nlm.nih.gov/pubmed/31610397
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.jpba.2019.112902
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