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Regulator of G-protein signaling (RGS) proteins as drug targets: Progress and future potentials

G protein–coupled receptors (GPCRs) play critical roles in regulating processes such as cellular homeostasis, responses to stimuli, and cell signaling. Accordingly, GPCRs have long served as extraordinarily successful drug targets. It is therefore not surprising that the discovery in the mid-1990s o...

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Pubblicato in:J Biol Chem
Autori principali: O'Brien, Joseph B., Wilkinson, Joshua C., Roman, David L.
Natura: Artigo
Lingua:Inglês
Pubblicazione: American Society for Biochemistry and Molecular Biology 2019
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6901330/
https://ncbi.nlm.nih.gov/pubmed/31636120
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.REV119.007060
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