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[b]-Annulated Halogen-Substituted Indoles as Potential DYRK1A Inhibitors

Since hyperactivity of the protein kinase DYRK1A is linked to several neurodegenerative disorders, DYRK1A inhibitors have been suggested as potential therapeutics for Down syndrome and Alzheimer’s disease. Most published inhibitors to date suffer from low selectivity against related kinases or from...

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Detalhes bibliográficos
Publicado no:Molecules
Main Authors: Lechner, Christian, Flaßhoff, Maren, Falke, Hannes, Preu, Lutz, Loaëc, Nadége, Meijer, Laurent, Knapp, Stefan, Chaikuad, Apirat, Kunick, Conrad
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2019
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6891749/
https://ncbi.nlm.nih.gov/pubmed/31766108
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules24224090
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