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Molecular dynamics simulations of aptamer-binding reveal generalized allostery in thrombin

Thrombin is an attractive target for antithrombotic therapy due to its central role in thrombosis and hemostasis as well as its role in inducing tumor growth, metastasis, and tumor invasion. The thrombin-binding DNA aptamer (TBA), is under investigation for anticoagulant drugs. Although aptamer bind...

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Dades bibliogràfiques
Publicat a:J Biomol Struct Dyn
Autors principals: Xiao, Jiajie, Salsbury, Freddie R.
Format: Artigo
Idioma:Inglês
Publicat: 2016
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6876308/
https://ncbi.nlm.nih.gov/pubmed/27794633
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1080/07391102.2016.1254682
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