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Tegavivint and the β-Catenin/ALDH Axis in Chemotherapy-Resistant and Metastatic Osteosarcoma

BACKGROUND: The Wnt/β-catenin pathway is closely associated with osteosarcoma (OS) development and metastatic progression. We investigated the antitumor activity of Tegavivint, a novel β-catenin/transducin β-like protein 1 (TBL1) inhibitor, against OS employing in vitro, ex vivo, and in vivo cell li...

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Podrobná bibliografie
Vydáno v:J Natl Cancer Inst
Hlavní autoři: Nomura, Motonari, Rainusso, Nino, Lee, Yi-Chien, Dawson, Brian, Coarfa, Cristian, Han, Ruolan, Larson, Jeffrey L, Shuck, Ryan, Kurenbekova, Lyazat, Yustein, Jason T
Médium: Artigo
Jazyk:Inglês
Vydáno: Oxford University Press 2019
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC6855956/
https://ncbi.nlm.nih.gov/pubmed/30793158
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1093/jnci/djz026
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