Cargando...

A Fluorescent Kinase Inhibitor that Exhibits Diagnostic Changes in Emission upon Binding

The development of a fluorescent LCK inhibitor that exhibits favourable solvatochromic properties upon binding the kinase is described. Fluorescent properties were realised through the inclusion of a prodan‐derived fluorophore into the pharmacophore of an ATP‐competitive kinase inhibitor. Fluorescen...

Descrición completa

Gardado en:
Detalles Bibliográficos
Publicado en:Angew Chem Int Ed Engl
Main Authors: Fleming, Cassandra L., Sandoz, Patrick A., Inghardt, Tord, Önfelt, Björn, Grøtli, Morten, Andréasson, Joakim
Formato: Artigo
Idioma:Inglês
Publicado: John Wiley and Sons Inc. 2019
Assuntos:
Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC6851755/
https://ncbi.nlm.nih.gov/pubmed/31411364
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/anie.201909536
Tags: Engadir etiqueta
Sen Etiquetas, Sexa o primeiro en etiquetar este rexistro!