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Preformulation and Evaluation of Tofacitinib as a Therapeutic Treatment for Asthma

Preformulation studies on tofacitinib citrate, a small molecule JAK3 specific inhibitor, have not been previously reported in literature. We therefore conducted several preformulation studies on tofacitinib citrate, and its free base, to better understand factors that affect its solubility, stabilit...

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Publicado en:AAPS PharmSciTech
Autores principales: Younis, Usir S., Vallorz, Ernest, Addison, Kenneth J., Ledford, Julie G., Myrdal, Paul B.
Formato: Artigo
Lenguaje:Inglês
Publicado: 2019
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC6818719/
https://ncbi.nlm.nih.gov/pubmed/30993508
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1208/s12249-019-1377-0
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