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Structural simplification: an efficient strategy in lead optimization

The trend toward designing large hydrophobic molecules for lead optimization is often associated with poor drug-likeness and high attrition rates in drug discovery and development. Structural simplification is a powerful strategy for improving the efficiency and success rate of drug design by avoidi...

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Bibliografski detalji
Izdano u:Acta Pharm Sin B
Glavni autori: Wang, Shengzheng, Dong, Guoqiang, Sheng, Chunquan
Format: Artigo
Jezik:Inglês
Izdano: Elsevier 2019
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC6804494/
https://ncbi.nlm.nih.gov/pubmed/31649841
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.apsb.2019.05.004
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