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OS4.2 Phase 0 trial of Ceritinib in brain metastasis and recurrent glioblastoma

BACKGROUND: Ceritinib is an orally bioavailable, small molecule inhibitor for ALK/IGFR1/FAK, which are highly expressed in glioblastoma and brain metastases. Preclinical and clinical data suggest that ceritinib has activity in central nervous system (CNS) malignancies, but to date there is no direct...

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Publicat a:Neuro Oncol
Autors principals: Fiorelli, R, Li, J, Bao, X, DeRogatis, A, Pennington-Krygier, C, Kim, S, Mehta, S, Sanai, N
Format: Artigo
Idioma:Inglês
Publicat: Oxford University Press 2019
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6795004/
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1093/neuonc/noz126.032
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