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A Phase 0 Trial of Ribociclib in Recurrent Glioblastoma Patients Incorporating a Tumor Pharmacodynamic- and Pharmacokinetic-Guided Expansion Cohort

BACKGROUND: CDK4/6-dependent cell-cycle regulation is disrupted in most glioblastomas. This study assesses the central nervous system (CNS) pharmacokinetics and tumor pharmacodynamics of ribociclib, a highly selective CDK4/6-inhibitor, in patients with recurrent glioblastoma. METHODS: Recurrent glio...

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Detalhes bibliográficos
Publicado no:Clin Cancer Res
Main Authors: Tien, An-Chi, Li, Jing, Bao, Xun, Derogatis, Alanna, Kim, Seongho, Mehta, Shwetal, Sanai, Nader
Formato: Artigo
Idioma:Inglês
Publicado em: 2019
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6863147/
https://ncbi.nlm.nih.gov/pubmed/31285369
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1158/1078-0432.CCR-19-0133
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