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Induction via Functional Protein Stabilization of Hepatic Cytochromes P450 upon gp78/Autocrine Motility Factor Receptor (AMFR) Ubiquitin E3-Ligase Genetic Ablation in Mice: Therapeutic and Toxicological Relevance

The hepatic endoplasmic reticulum (ER)–anchored monotopic proteins, cytochromes P450 (P450s), are enzymes that metabolize endobiotics (physiologically active steroids and fatty acids), as well as xenobiotics including therapeutic/chemotherapeutic drugs, nutrients, carcinogens, and toxins. Alteration...

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Publicado en:Mol Pharmacol
Autores principales: Kwon, Doyoung, Kim, Sung-Mi, Jacob, Peyton, Liu, Yi, Correia, Maria Almira
Formato: Artigo
Lenguaje:Inglês
Publicado: The American Society for Pharmacology and Experimental Therapeutics 2019
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC6790065/
https://ncbi.nlm.nih.gov/pubmed/31492698
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.119.117069
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