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Does the Lipid Bilayer Orchestrate Access and Binding of Ligands to Transmembrane Orthosteric/Allosteric Sites of G Protein-Coupled Receptors?

The ligand-binding sites of many G protein-coupled receptors (GPCRs) are situated around and deeply embedded within the central pocket formed by their seven transmembrane-spanning α-helical domains. Generally, these binding sites are assumed accessible to endogenous ligands from the aqueous phase. R...

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Détails bibliographiques
Publié dans:Mol Pharmacol
Auteurs principaux: Szlenk, Christopher T., GC, Jeevan B., Natesan, Senthil
Format: Artigo
Langue:Inglês
Publié: The American Society for Pharmacology and Experimental Therapeutics 2019
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC6776015/
https://ncbi.nlm.nih.gov/pubmed/30967440
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.118.115113
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