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Site Selective Antibody-Oligonucleotide Conjugation via Microbial Transglutaminase

Nucleic Acid Therapeutics (NATs), including siRNAs and AntiSense Oligonucleotides (ASOs), have great potential to drug the undruggable genome. Targeting siRNAs and ASOs to specific cell types of interest has driven dramatic improvement in efficacy and reduction in toxicity. Indeed, conjugation of tr...

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Détails bibliographiques
Publié dans:Molecules
Auteurs principaux: Huggins, Ian J., Medina, Carlos A., Springer, Aaron D., van den Berg, Arjen, Jadhav, Satish, Cui, Xianshu, Dowdy, Steven F.
Format: Artigo
Langue:Inglês
Publié: MDPI 2019
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC6767100/
https://ncbi.nlm.nih.gov/pubmed/31509944
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules24183287
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