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Construction of a Fluorescent Screening System of Allosteric Modulators for the GABA(A) Receptor Using a Turn-On Probe

[Image: see text] γ-Aminobutyric acid (GABA) is the major inhibitory neurotransmitter in the central nervous system. The fast inhibitory actions of GABA are mainly mediated by GABA(A) receptors (GABA(A)Rs), which are widely recognized as clinically relevant drug targets. However, it remains difficul...

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Argitaratua izan da:ACS Cent Sci
Egile Nagusiak: Sakamoto, Seiji, Yamaura, Kei, Numata, Tomohiro, Harada, Fumio, Amaike, Kazuma, Inoue, Ryuji, Kiyonaka, Shigeki, Hamachi, Itaru
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: American Chemical Society 2019
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC6764212/
https://ncbi.nlm.nih.gov/pubmed/31572781
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acscentsci.9b00539
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