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Functional characteristics of CYP3A4 allelic variants on the metabolism of loperamide in vitro

BACKGROUND: Cytochrome P450 3A4 (CYP3A4) appears to be genetically polymorphic, which in turn contributes to interindividual variability in response to therapeutic drugs. Loperamide, identified as a CYP3A4 substrate, is prone to misuse and abuse and has high risks of life-threatening cardiotoxicity....

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Publicat a:Infect Drug Resist
Autors principals: Lin, Qian-Meng, Li, Ying-Hui, Liu, Qian, Pang, Ni-Hong, Xu, Ren-Ai, Cai, Jian-Ping, Hu, Guo-Xin
Format: Artigo
Idioma:Inglês
Publicat: Dove 2019
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6750855/
https://ncbi.nlm.nih.gov/pubmed/31571937
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.2147/IDR.S215129
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