Llwytho...

Targeted Rediscovery and Biosynthesis of the Farnesyl-Transferase Inhibitor Pepticinnamin E

The natural product pepticinnamin E potently inhibits protein farnesyl transferases and has potential applications in treating cancer and malaria. Pepticinnamin E contains a rare N-terminal cinnamoyl moiety and several nonproteinogenic amino acids including an unusual 2-chloro-4-O-methyl-3,4-dihydro...

Disgrifiad llawn

Wedi'i Gadw mewn:
Manylion Llyfryddiaeth
Cyhoeddwyd yn:Chembiochem
Prif Awduron: Maria, Kevin C. Santa, Chan, Andrew N., O’Neill, Erinn M., Li, Bo
Fformat: Artigo
Iaith:Inglês
Cyhoeddwyd: 2019
Pynciau:
Mynediad Ar-lein:https://ncbi.nlm.nih.gov/pmc/articles/PMC6750724/
https://ncbi.nlm.nih.gov/pubmed/30694017
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cbic.201900025
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