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Unexpected Mutations in HIV-1 That Confer Resistance to the Tat Inhibitor Didehydro-Cortistatin A

Didehydro-cortistatin A (dCA) is a human immunodeficiency virus type 1 (HIV-1) Tat inhibitor that functions by selectively binding to the RNA binding domain of Tat. In addition to inhibiting viral replication, dCA can drive HIV-1 into a state of “deep latency” in which latent viruses are refractory...

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Pubblicato in:mBio
Autore principale: Rice, Andrew P.
Natura: Artigo
Lingua:Inglês
Pubblicazione: American Society for Microbiology 2019
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6747727/
https://ncbi.nlm.nih.gov/pubmed/31289189
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/mBio.01547-19
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