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Structural Insights into the Interaction of Cytochrome P450 3A4 with Suicide Substrates: Mibefradil, Azamulin and 6′,7′-Dihydroxybergamottin

Human cytochrome P450 3A4 (CYP3A4) is the most important drug-metabolizing enzyme. Some drugs and natural compounds can act as suicide (mechanism-based) inactivators of CYP3A4, leading to unanticipated drug-drug interactions, toxicity and therapeutic failures. Despite significant clinical and toxico...

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Bibliografiske detaljer
Udgivet i:Int J Mol Sci
Hovedforfatter: Sevrioukova, Irina F.
Format: Artigo
Sprog:Inglês
Udgivet: MDPI 2019
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC6747129/
https://ncbi.nlm.nih.gov/pubmed/31480231
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms20174245
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