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Extrasynaptic GABA(A) Receptors of Thalamocortical Neurons: A Molecular Target for Hypnotics

Among hypnotic agents that enhance GABA(A) receptor function, etomidate is unusual because it is selective for β(2)/β(3) compared with β(1) subunit-containing GABA(A) receptors. Mice incorporating an etomidate-insensitive β(2) subunit (β(2N265S)) revealed that β(2) subunit-containing receptors media...

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Dades bibliogràfiques
Publicat a:J Neurosci
Autors principals: Belelli, Delia, Peden, Dianne R., Rosahl, Thomas W., Wafford, Keith A., Lambert, Jeremy J.
Format: Artigo
Idioma:Inglês
Publicat: Society for Neuroscience 2005
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6726038/
https://ncbi.nlm.nih.gov/pubmed/16354909
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1523/JNEUROSCI.2679-05.2005
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