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ADME Considerations and Bioanalytical Strategies for Pharmacokinetic Assessments of Antibody-Drug Conjugates

Antibody-drug conjugates (ADCs) are a unique class of biotherapeutics of inherent heterogeneity and correspondingly complex absorption, distribution, metabolism, and excretion (ADME) properties. Herein, we consider the contribution of various components of ADCs such as various classes of warheads, l...

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Detalhes bibliográficos
Publicado no:Antibodies (Basel)
Main Authors: Mou, Si, Huang, Yue, Rosenbaum, Anton I.
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2018
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6698957/
https://ncbi.nlm.nih.gov/pubmed/31544891
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/antib7040041
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