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Structural basis of lysosomal phospholipase A(2) inhibition by Zn(2+)

Lysosomal phospholipase A(2) (LPLA(2)/PLA2G15) is a key enzyme involved in lipid homeostasis and is characterized by both phospholipase A2 and transacylase activity, and an acidic pH optimum. Divalent cations such as Ca(2+) and Mg(2+) have previously been shown to have little effect on the activity...

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Publicat a:Biochemistry
Autors principals: Bouley, Renee A., Hinkovska-Galcheva, Vania, Shayman, James A., Tesmer, John J. G.
Format: Artigo
Idioma:Inglês
Publicat: 2019
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6677152/
https://ncbi.nlm.nih.gov/pubmed/30830753
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.biochem.8b01124
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