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Conservation of Potentially Druggable Cavities in Intrinsically Disordered Proteins

[Image: see text] Intrinsically disordered proteins (IDPs) exist in highly dynamic conformational ensembles, which pose a major obstacle for drug development targeting IDPs because traditional rational drug design relies on unique three-dimensional structures. Here, we analyzed the conservation (esp...

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Detalhes bibliográficos
Publicado no:ACS Omega
Main Authors: Chong, Bin, Li, Maodong, Li, Tong, Yu, Miao, Zhang, Yugang, Liu, Zhirong
Formato: Artigo
Idioma:Inglês
Publicado em: American Chemical Society 2018
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6643371/
https://ncbi.nlm.nih.gov/pubmed/31458221
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsomega.8b02092
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