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Non-nucleoside Reverse Transcriptase Inhibitors Inhibit Reverse Transcriptase through a Mutually Exclusive Interaction with Divalent Cation-dNTP Complexes

Non-nucleoside reverse transcriptase inhibitors (NNRTIs) are considered noncompetitive inhibitors that structurally alter reverse transcriptase (RT) and dramatically decrease catalysis. In this report, biochemical analysis with various divalent cations was used to demonstrate that NNRTIs and divalen...

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Dettagli Bibliografici
Pubblicato in:Biochemistry
Autore principale: DeStefano, Jeffrey J.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2019
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6629025/
https://ncbi.nlm.nih.gov/pubmed/30900874
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.biochem.9b00028
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