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Ranking Reversible Covalent Drugs: From Free Energy Perturbation to Fragment Docking

Reversible covalent inhibitors have drawn increasing attention in drug design, as they are likely more potent than noncovalent inhibitors and less toxic than covalent inhibitors. Despite those advantages, the computational prediction of reversible covalent binding presents a formidable challenge bec...

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Détails bibliographiques
Publié dans:J Chem Inf Model
Auteurs principaux: Zhang, Han, Jiang, Wenjuan, Chatterjee, Payal, Luo, Yun
Format: Artigo
Langue:Inglês
Publié: 2019
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC6610880/
https://ncbi.nlm.nih.gov/pubmed/30763080
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jcim.8b00959
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