Загрузка...

The L46P Mutant Confers a Novel Allosteric Mechanism of Resistance Toward the Influenza A Virus M2 S31N Proton Channel Blockers

The Food and Drug Administration–approved influenza A antiviral amantadine inhibits the wild-type (WT) AM2 channel but not the S31N mutant predominantly found in circulating strains. In this study, serial viral passages were applied to select resistance against a newly developed isoxazole-conjugated...

Полное описание

Сохранить в:
Библиографические подробности
Опубликовано в: :Mol Pharmacol
Главные авторы: Musharrafieh, Rami, Lagarias, Panagiotis I., Ma, Chunlong, Tan, Gene S., Kolocouris, Antonios, Wang, Jun
Формат: Artigo
Язык:Inglês
Опубликовано: The American Society for Pharmacology and Experimental Therapeutics 2019
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC6608606/
https://ncbi.nlm.nih.gov/pubmed/31175183
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.119.116640
Метки: Добавить метку
Нет меток, Требуется 1-ая метка записи!