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Calculate Protein-Ligand Binding Affinities with the Extended Linear Interaction Energy Method: Application on the Cathepsin S Set in the D3R Grand Challenge 3

We participated the Cathepsin S (CatS) sub-challenge of the Drug Design Data Resource (D3R) Grand Challenge 3 (GC3) in 2017 to blindly predict the binding poses of 24 CatS-bound ligands, the binding affinity ranking of 136 ligands, and the binding free energies of a subset of 33 ligands in Stage 1A...

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Dettagli Bibliografici
Pubblicato in:J Comput Aided Mol Des
Autori principali: HE, Xibing, MAN, Viet H., JI, Beihong, XIE, Xiang-Qun, WANG, Junmei
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2018
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6608581/
https://ncbi.nlm.nih.gov/pubmed/30218199
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s10822-018-0162-6
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