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Experimental and Computational Studies Delineate the Role of Asparagine 177 in Hydride Transfer for E. coli Thymidylate Synthase

Thymidylate synthase (TSase), an enzyme responsible for the de novo biosynthesis of 2’-deoxythymidine 5’-monophosphate (thymidylate, dTMP) necessary for DNA synthesis, has been a drug target for decades. TSase is a highly conserved enzyme across species ranging from very primitive organisms to mamma...

Täydet tiedot

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Bibliografiset tiedot
Julkaisussa:ACS Catal
Päätekijät: Gurevic, Ilya, Islam, Zahidul, Świderek, Katarzyna, Trepka, Kai, Ghosh, Ananda K., Moliner, Vicent, Kohen, Amnon
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: 2018
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC6605054/
https://ncbi.nlm.nih.gov/pubmed/31275729
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acscatal.8b02554
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