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Molecular mechanisms of human P2X3 receptor channel activation and modulation by divalent cation bound ATP

P2X3 receptor channels expressed in sensory neurons are activated by extracellular ATP and serve important roles in nociception and sensory hypersensitization, making them attractive therapeutic targets. Although several P2X3 structures are known, it is unclear how physiologically abundant Ca(2+)-AT...

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Dettagli Bibliografici
Pubblicato in:eLife
Autori principali: Li, Mufeng, Wang, Yao, Banerjee, Rahul, Marinelli, Fabrizio, Silberberg, Shai, Faraldo-Gómez, José D, Hattori, Motoyuki, Swartz, Kenton Jon
Natura: Artigo
Lingua:Inglês
Pubblicazione: eLife Sciences Publications, Ltd 2019
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6590987/
https://ncbi.nlm.nih.gov/pubmed/31232692
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.7554/eLife.47060
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