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Systemic Design and Evaluation of Ticagrelor-Loaded Nanostructured Lipid Carriers for Enhancing Bioavailability and Antiplatelet Activity

Ticagrelor (TGL), a P2Y(12) receptor antagonist, is classified as biopharmaceutics classification system (BCS) class IV drug due to its poor solubility and permeability, resulting in low oral bioavailability. Nanostructured lipid carriers (NLC) are an efficient delivery system for the improvement of...

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Detalhes bibliográficos
Publicado no:Pharmaceutics
Main Authors: Son, Gi-Ho, Na, Young-Guk, Huh, Hyun Wook, Wang, Miao, Kim, Min-Ki, Han, Min-Gu, Byeon, Jin-Ju, Lee, Hong-Ki, Cho, Cheong-Weon
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2019
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6572397/
https://ncbi.nlm.nih.gov/pubmed/31071977
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/pharmaceutics11050222
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