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Syntheses and in vitro biological evaluation of S1PR1 ligands and PET studies of four F-18 labeled radiotracers in the brain of nonhuman primates

A series of seventeen hydroxyl-containing sphingosine 1-phosphate receptor 1 (S1PR1) ligands were designed and synthesized. Their in vitro binding potencies were determined using [(32)P]S1P competitive binding assays. Compounds 10a, 17a, 17b, and 24 exhibited high S1PR1 binding potencies with IC(50)...

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Vydáno v:Org Biomol Chem
Hlavní autoři: Luo, Zonghua, Han, Junbin, Liu, Hui, Rosenberg, Adam J., Chen, Delphine L., Gropler, Robert J., Perlmutter, Joel S., Tu, Zhude
Médium: Artigo
Jazyk:Inglês
Vydáno: 2018
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC6561338/
https://ncbi.nlm.nih.gov/pubmed/30462126
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c8ob02609b
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