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Inhibition of β-catenin/B cell lymphoma 9 protein−protein interaction using α-helix–mimicking sulfono-γ-AApeptide inhibitors

The rational design of α-helix–mimicking peptidomimetics provides a streamlined approach to discover potent inhibitors for protein−protein interactions (PPIs). However, designing cell-penetrating long peptidomimetic scaffolds equipped with various functional groups necessary for interacting with lar...

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Publicado en:Proc Natl Acad Sci U S A
Autores principales: Sang, Peng, Zhang, Min, Shi, Yan, Li, Chunpu, Abdulkadir, Sami, Li, Qi, Ji, Haitao, Cai, Jianfeng
Formato: Artigo
Lenguaje:Inglês
Publicado: National Academy of Sciences 2019
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC6561201/
https://ncbi.nlm.nih.gov/pubmed/31088961
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.1819663116
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