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Sustained delivery of a camptothecin prodrug – CZ48 by nanosuspensions with improved pharmacokinetics and enhanced anticancer activity

Background and aim: We have synthesized a novel lactone-stabilized camptothecin (CPT) analog named CZ48 and demonstrated its potent anticancer effects via bioconversion to the active CPT in earlier studies. Herein, we aimed to develop, optimize and characterize CZ48 nanosuspensions, for a sustained...

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Detalhes bibliográficos
Publicado no:Int J Nanomedicine
Main Authors: Dong, Dong, Hsiao, Cheng-Hui, Giovanella, Beppino C, Wang, Yifei, Chow, Diana SL, Li, Zhijie
Formato: Artigo
Idioma:Inglês
Publicado em: Dove 2019
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6540077/
https://ncbi.nlm.nih.gov/pubmed/31213802
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.2147/IJN.S196453
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