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In Vitro and In Vivo Efficacy of the Monocarboxylate Transporter 1 Inhibitor AR-C155858 in the Murine 4T1 Breast Cancer Tumor Model

Monocarboxylate transporter 1 (MCT1), also known as a l-lactate transporter, is a potential therapeutic target in cancer. The objectives of this study were to evaluate efficacy and assess concentration-effect relationships of AR-C155858 (a selective and potent MCT1 inhibitor) in murine 4T1 breast ca...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Argitaratua izan da:AAPS J
Egile Nagusiak: Guan, Xiaowen, Bryniarski, Mark A., Morris, Marilyn E.
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: 2018
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC6536115/
https://ncbi.nlm.nih.gov/pubmed/30397860
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1208/s12248-018-0261-2
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