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Tolerance to WIN55,212-2 is delayed in desensitization-resistant S426A/S430A mice

Tolerance to cannabinoid agonists can develop through desensitization of the cannabinoid receptor 1 (CB(1)) following prolonged administration. Desensitization results from phosphorylation of CB(1) by a G protein-coupled receptor kinase (GRK), and subsequent association of the receptor with arrestin...

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Publicado en:Neuropharmacology
Autores principales: Nealon, Caitlin M., Henderson-Redmond, Angela N., Hale, David E., Morgan, Daniel J.
Formato: Artigo
Lenguaje:Inglês
Publicado: 2019
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC6535342/
https://ncbi.nlm.nih.gov/pubmed/30629988
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.neuropharm.2018.12.026
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