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Studies Towards Hypoxia-Activated Prodrugs of PARP Inhibitors

Poly(ADP-ribose)polymerase (PARP) inhibitors (PARPi) have recently been approved for the treatment of breast and ovarian tumors with defects in homologous recombination repair (HRR). Although it has been demonstrated that PARPi also sensitize HRR competent tumors to cytotoxic chemotherapies or radio...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Argitaratua izan da:Molecules
Egile Nagusiak: Dickson, Benjamin D., Wong, Way Wua, Wilson, William R., Hay, Michael P.
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: MDPI 2019
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC6514732/
https://ncbi.nlm.nih.gov/pubmed/31010230
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules24081559
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