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Semisynthetic Analogues of Anhydrotetracycline as Inhibitors of Tetracycline Destructase Enzymes

The synthesis and biological evaluation of semisynthetic anhydrotetracycline analogues as small molecule inhibitors of tetracycline-inactivating enzymes are reported. Inhibitor potency was found to vary as a function of enzyme (major) and substrate-inhibitor pair (minor), and anhydrotetracycline ana...

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Vydáno v:ACS Infect Dis
Hlavní autoři: Markley, Jana L., Fang, Luting, Gasparrini, Andrew J., Symister, Chanez T., Kumar, Hirdesh, Tolia, Niraj H., Dantas, Gautam, Wencewicz, Timothy A.
Médium: Artigo
Jazyk:Inglês
Vydáno: 2019
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On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC6490184/
https://ncbi.nlm.nih.gov/pubmed/30835428
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsinfecdis.8b00349
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