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V1 and V2 Domains of HIV Envelope Contribute to CCR5 Antagonist Resistance

Vicriviroc (VCV) is a CCR5 antagonist that blocks the viral entry of CCR5-tropic (R5) virions by binding to and inducing a conformational change in the chemokine receptor. Clinical resistance to CCR5 antagonists occurs in two phases, competitive and noncompetitive stages. In this study, we analyzed...

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Detalles Bibliográficos
Publicado en:J Virol
Autores principales: Wu, Ellen, Du, Yueqi, Gao, Xiang, Zhang, Jie, Martin, John, Mitreva, Makedonka, Ratner, Lee
Formato: Artigo
Lenguaje:Inglês
Publicado: American Society for Microbiology 2019
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC6475789/
https://ncbi.nlm.nih.gov/pubmed/30787151
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/JVI.00050-19
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