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Diarylcarbonates are a new class of deubiquitinating enzyme inhibitors

Promiscuous inhibitors of tyrosine protein kinases, proteases and phosphatases are useful reagents for probing regulatory pathways and stabilizing lysates as well as starting points for the design of more targeted agents. Ubiquitination regulates many critical cellular processes, and promiscuous inh...

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Dades bibliogràfiques
Publicat a:Bioorg Med Chem Lett
Autors principals: Long, Marcus J. C., Lawson, Ann P., Baggio, Rick, Qian, Yu, Rozhansky, Lior, Fasci, Domenico, Oualid, Farid El, Weerapana, Eranthie, Hedstrom, Lizbeth
Format: Artigo
Idioma:Inglês
Publicat: 2018
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6467287/
https://ncbi.nlm.nih.gov/pubmed/30528168
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2018.11.055
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