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Diarylcarbonates are a new class of deubiquitinating enzyme inhibitors

Promiscuous inhibitors of tyrosine protein kinases, proteases and phosphatases are useful reagents for probing regulatory pathways and stabilizing lysates as well as starting points for the design of more targeted agents. Ubiquitination regulates many critical cellular processes, and promiscuous inh...

Täydet tiedot

Tallennettuna:
Bibliografiset tiedot
Julkaisussa:Bioorg Med Chem Lett
Päätekijät: Long, Marcus J. C., Lawson, Ann P., Baggio, Rick, Qian, Yu, Rozhansky, Lior, Fasci, Domenico, Oualid, Farid El, Weerapana, Eranthie, Hedstrom, Lizbeth
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: 2018
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC6467287/
https://ncbi.nlm.nih.gov/pubmed/30528168
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2018.11.055
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