Caricamento...

Bruton's tyrosine kinase (Btk) inhibitor tirabrutinib suppresses osteoclastic bone resorption

Osteoclasts are responsible for bone erosion in osteoporosis and rheumatoid arthritis (RA). Both Btk and Tec kinases have essential functions in osteoclast differentiation. Tirabrutinib is a highly potent and dual oral Btk/Tec inhibitor with an IC(50) in the nmol/L range and significantly inhibits t...

Descrizione completa

Salvato in:
Dettagli Bibliografici
Pubblicato in:Bone Rep
Autori principali: Ariza, Yuko, Murata, Masayuki, Ueda, Yoshiko, Yoshizawa, Toshio
Natura: Artigo
Lingua:Inglês
Pubblicazione: Elsevier 2019
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6431727/
https://ncbi.nlm.nih.gov/pubmed/30956999
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bonr.2019.100201
Tags: Aggiungi Tag
Nessun Tag, puoi essere il primo ad aggiungerne! !