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Carbonic anhydrase II in complex with carboxylic acid-based inhibitors

Carbonic anhydrases (CAs) are molecular targets in various diseases. While many sulfonamide-based drugs are in clinical use, CA inhibitor design is moving towards the incorporation of alternative zinc-binding groups, such as carboxylic acids, to promote CA isoform-specific inhibition. Here, X-ray cr...

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Detalhes bibliográficos
Publicado no:Acta Crystallogr F Struct Biol Commun
Main Authors: Lomelino, Carrie L., McKenna, Robert
Formato: Artigo
Idioma:Inglês
Publicado em: International Union of Crystallography 2019
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6404860/
https://ncbi.nlm.nih.gov/pubmed/30839290
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1107/S2053230X18018344
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